Chingerezi: Odiganan
Nambala ya Cas: 204248-72-27-27-27-27-27-27-27-27
Njira ya molecular: C₉₀h₁₂₇n₂₇o₁₂
Kulemera kwa maselo: 1779.15
Mndandanda: Ilrwpwwpwrrk-nh2
Maonekedwe: oyera kapena oyera-ufa
Momwe Osiganan amachita:
Ndi peptide yaying'ono kwambiri ndipo chifukwa chake imavuta kuzindikira ndikulemba mapulojekiti; Imakhala yokhazikika pa cermiyu kuti muthe kukana purteyolysis ndikuchotsa chikwangwani cha Carboxyl. It is amphiphilic and can interact strongly with the cell membrane. Cell membrane akuyembekezeka kukhala imodzi mwazinthu zazikulu. Ndi polycation yomwe imakondweretsa kuyanjana kwawo ndi bacrateria ndi zitsamba zakunja za Lipolyulsaride (LPS) ndi peptidoglycan. Mu mabakiteriya, kuthekera kwa membrane kumakhala kovuta kwambiri kuposa maselo a anthu akumali, omwe amatha kukulitsa ma bantibiotian ndi kutumiza. Chochititsa chomaliza ndi chilema champhamvu chomwe antiinflammination chomwe antiminidina adagwiranso ntchito pa erythrocyte, pomwe Odiganan akuwoneka kuti sakhala ndi hemolyte. As mentioned above, the charged residues of omiga-nan are located near each terminal, away from the central hydrophobic region of the peptide, and the total positive charge of the peptide increases from 4+ to 5+, which can be explained by reduced hemolysis, since these changes are not favorable for peptide-like substances associated with zwitt-rionic mammalian membranes. Izi zimathandizidwa ndi zotsatira za kuphulika ndi ena, pomwe chidutswa chapakati cha kupindika kwa antiinflamlat chimalumikizidwa ndi ntchito, pomwe chidutswa cholumikizira chikuwoneka kuti chikusintha mawonekedwe a chandamale.
Odiganan amagwiritsidwa ntchito:
Odiganan ndi njira yopanga cholumikizira coptic tepipde pakali pano poyambitsa matenda okhudzana ndi Catheter ndi chithandizo cha ziphuphu ndi rosacea. Mu kafukufukuyu, tinkayesa kuchita bwino kwambiri kwa Odiganan gel ozungulira pakhungu ziwiri (ku Viva Porcine khungu la nkhumba komanso khungu la nkhumba). Odiganan0 adayesedwa mu mtundu wa Ex Viva Porcne Corcroniation Plannation 1 mpaka 2% ya gl wa gl Panalibe kusiyana kwakukulu mu zochitika pakati pa meticillin-pormphycocccus ndi astrackcocccus a Aureus Aureus, ndi mankhwala osokoneza bongo sanakhudzidwe ndi kukula kwa chinthu chomwe chapezeka. Odiganan1% Geli anali ndi mankhwala a antificrobial radickari, yochepetsa (10) mu magawo 10) a staphylococcus epidelmolis / tsamba pa Flagella / Tsamba 24 H pambuyo pa ntchito. Ntchito ya antibacterial ndi antifungal ntchito ya odiganan1% yotsimikizika idatsimikiziridwa ndi kafukufuku wina mu mtundu wa khungu la dolphin. Mwachidule, ma gels am'miganem awonetsedwa kuti ali ndi matenda a bactericidal komanso bactericidal omwe ali ndi vuto lodalira kwambiri pamlingo wowoneka bwino. Zotsatira izi zimawonetsanso kuthekera kwa mankhwalawa ngati antimicicrobial wothandizira.
Post Nthawi: 2025-07-02