chiyambi
Goretide, omwe amadziwikanso kuti n-acetyl-serine - aspartic acid - proline - tetter-lys-lys-lys-ac-ng-d-d-d-d-rolicle - madzi amthupi osiyanasiyana m'thupi. Tetrapeptide iyi imamasulidwa ndi Prolyl oligoptedase (pop), yomwe imayambitsidwa ndi pymosin yake. Kukhazikika kwa magazi nthawi zambiri kumakhala pa sikelo ya nanomole.
makupalat
Malinga ndi kafukufuku wa pharmacokinetic ya goretidide, pambuyo pa jakisoni wamkati, goretilaude mwachangu zimasokonekera ndi theka la moyo wa 4 ~ 5min. Greretitide idayeretsedwa ndi plasma ya anthu mwa njira ziwiri: ① Angiotensin-kutembenuza enzyme (Ace)-hydrolysis; ② Kuwonjezeka kwa glomerlar. Hydrolysis wa angiotensin kusintha enzyme (Ace) ndiye njira yayikulu ya kagayidwe kambiri.
Zochita Zachilengedwe
Goretitide ndi mtundu wa zowongolera zowongolera zowongolera zomwe zimapangidwa ndi zinthu zosiyanasiyana zachilengedwe. Zinali zisanachitike kuti a Greretide akhoza kuletsa kulowa kwa maselo oyamba a hematopopoietic. Pambuyo pake adapezeka kuti a Greretide amatha kusintha kuthekera kolimbikitsa mapangidwe am'magazi ndikuthandizira kuchiritsa kwa zilonda m'malonda owonongeka. Goretitide imatha kuletsa kusiyanitsa kwa mafupa am'mimba maselo omwe amalimbikitsidwa ndi mgm kukhala macrophages, motero amasewera ndi kutupa. Goretitide yapezeka posachedwa kuti ilepheretse kuchuluka kwa maselo osiyanasiyana.
gwilitsa nchito
Monga polypeptide zinthu, goretide angagwiritsidwe ntchito ngati mankhwala osokoneza bongo.
Post Nthawi: 2025-07-03